OpenLegislation

Regulation (EU) No 1238/2010 of the European Parliament and of the Council of 15 December 2010 amending Annex I to Council Regulation (EEC) No 2658/87 as regards the provision of duty-free treatment for specified pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organization and specified products used for the manufacture of finished pharmaceuticals

EU Regulation No 1238/2010 · Adopted 15 December 2010 · Extends to United Kingdom

Original text. legislation.gov.uk does not revise this item, so later amendments are not shown here. Changes made to it are listed under each provision when known.

Regulation (EU) No 1238/2010 of the European Parliament and of the Council

of 15 December 2010

amending Annex I to Council Regulation (EEC) No 2658/87 as regards the provision of duty-free treatment for specified pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organization and specified products used for the manufacture of finished pharmaceuticals

THE EUROPEAN PARLIAMENT AND THE COUNCIL OF THE EUROPEAN UNION,

Having regard to the Treaty on the Functioning of the European Union, and in particular Article 207 thereof,

Having regard to the proposal from the European Commission,

After transmission of the draft legislative act to the national parliaments,

Acting in accordance with the ordinary legislative proceduref1,

Whereas:

(1)

In the course of the Uruguay Round negotiations, the Community and a number of countries agreed that duty-free treatment should be granted to pharmaceutical products falling within the Harmonised System (HS) Chapter 30 and HS headings 2936, 2937, 2939 and 2941 as well as to designated pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organization, specified salts, esters and hydrates of such INNs, and designated pharmaceutical intermediates used for the production and manufacture of finished pharmaceuticals.

(2)

The results of the discussions, as set out in the Record of Discussions, were incorporated into the tariff schedules of the participants annexed to the Marrakesh Protocol to the General Agreement on Tariffs and Trade (GATT) 1994.

(3)

Participants concluded that representatives of World Trade Organization (WTO) members, party to the Record of Discussions, would meet under the auspices of the Council for Trade in Goods of the WTO, normally at least once every three years, to review the product coverage with a view to including, by consensus, additional pharmaceutical products for tariff elimination.

(4)

Three such reviews have taken place with the result that a certain number of additional INNs and pharmaceutical intermediates used for the production and manufacture of finished pharmaceuticals have been granted duty-free treatment, that some of those intermediates have been transferred to the list of INNs, and that the list of specified prefixes and suffixes for salts, esters or hydrates of INNs has been expanded.

(5)

A fourth review was deemed appropriate and was launched in 2009. It concluded that a certain number of additional INNs and pharmaceutical intermediates used for the production and manufacture of finished pharmaceuticals should be granted duty-free treatment, that some of those intermediates already included in the pharmaceutical sectoral arrangement and its revisions should be transferred to the list of INNs, and that the list of specified prefixes and suffixes for salts, esters or hydrates of INNs should be expanded.

(6)

Council Regulation (EEC) No 2658/87 of 23 July 1987 on the tariff and statistical nomenclature and on the Common Customs Tarifff2 established the Combined Nomenclature (CN) and set out the conventional duty rates of the Common Customs Tariff.

(7)

Regulation (EEC) No 2658/87 should therefore be amended accordingly.

(8)

In order to ensure that the measures provided for in this Regulation apply from 1 January 2011, it should enter into force on the day following that of its publication,

HAVE ADOPTED THIS REGULATION:

Annotations to the whole text

Footnotes

f1

Position of the European Parliament of 23 November 2010 (not yet published in the Official Journal) and decision of the Council of 10 December 2010.

f2

OJ L 256, 7.9.1987, p. 1.

Contents

  1. 1Article 1
  2. 2Article 2
  3. Signature
  4. Annex IAnnex I
  5. Annex IIList of prefixes and suffixes which, in combination with the INNs of Annex 3 to Annex I to Regulation (EEC) No 2658/87, describe the salts, esters or hydrates of INNs; these salts, esters and hydrates are free of duty, on condition that they are classifiable in the same six-digit HS subheading as the corresponding INN
  6. Annex IIIAnnex III
  7. Annex IVAnnex IV

1

Annexes 3, 4 and 6 of Section II of Part Three of Annex I to Regulation (EEC) No 2658/87 (Lists of pharmaceutical substances which qualify for duty-free treatment) are hereby amended as follows:

  1. 1..

    As from 1 January 2011 the Union shall extend duty-free treatment to the INNs listed in Annex I.

  2. 2..

    As from 1 January 2011 the list of prefixes and suffixes which, in combination with the INNs included in the pharmaceutical sectoral arrangement and its revisions, describe the salts, esters or hydrates of INNs which are also eligible for duty-free treatment, on condition that they are classifiable in the same six-digit HS subheading as the corresponding INN, shall be amended as set out in Annex II.

  3. 3..

    As from 1 January 2011 the Union shall extend duty-free treatment to the pharmaceutical intermediates used in the production and manufacture of finished pharmaceuticals, listed in Annex III.

  4. 4..

    As from 1 January 2011 the pharmaceutical intermediates listed in Annex IV shall be withdrawn from the list of such compounds receiving duty-free treatment.

2

This Regulation shall enter into force on the day following that of its publication in the Official Journal of the European Union.

It shall apply from 1 January 2011.

Signature

This Regulation shall be binding in its entirety and directly applicable in all Member States.

Done at Strasbourg, 15 December 2010.

For the European Parliament

The President

J. Buzek

For the Council

The President

O. Chastel

Annex I

List of international non-proprietary names (INNs) to be added to the list of products receiving duty-free treatment included in Annex 3 to Annex I to Regulation (EEC) No 2658/87

CN codeCAS RNName
2842 90 80 119175-48-3fermagate
2843 90 90 759457-82-4padeliporfin
2844 40 30 123748-56-1iodofiltic acid ( 123 I )
2904 10 00 21668-77-9eprodisate
2906 19 00 199798-84-0elocalcitol
2909 30 90 24150-24-1terameprocol
2916 19 95 81485-25-8peretinoin
2916 39 00 51543-40-9tarenflurbil
2918 19 98 174022-42-5bevirimat
2919 90 00 258516-89-1fospropofol
2920 90 85 163133-43-5naproxcinod
2921 19 99 3687-18-1tramiprosate
2922 19 85 68392-35-8afimoxifene
2922 19 85 753449-67-1ronacaleret
2922 29 00 433265-65-7faxeladol
2922 50 00 121524-08-1amibegron
2922 50 00 329773-35-5cinaciguat
2922 50 00 643094-49-9fasobegron
2923 10 00 856676-23-8choline fenofibrate
2924 29 98 847353-30-4arbaclofen placarbil
2924 29 98 194785-19-8bedoradrine
2924 29 98 194085-75-1carisbamate
2924 29 98 254750-02-2emricasan
2924 29 98 355129-15-6eprotirome
2924 29 98 402567-16-2firategrast
2924 29 98 478296-72-9gabapentin enacarbil
2924 29 98 15866-90-7incyclinide
2924 29 98 202844-10-8indantadol
2924 29 98 96847-55-1levomilnacipran
2924 29 98 608137-32-2lisdexamfetamine
2924 29 98 652990-07-3milveterol
2924 29 98 181816-48-8ombrabulin
2924 29 98 289656-45-7senicapoc
2925 19 95 19171-19-8pomalidomide
2928 00 90 22033-87-0olesoxime
2928 00 90 2675-35-6sivifene
2928 00 90 816458-31-8tecovirimat
2928 00 90 238750-77-1tosedostat
2928 00 90 149647-78-9vorinostat
2929 90 00 31645-39-3palifosfamide
2930 90 99 608141-41-9apremilast
2930 90 99 216167-92-9camobucol
2930 90 99 211513-37-0dalcetrapib
2930 90 99 69819-86-9darinaparsin
2930 90 99 488832-69-5elesclomol
2930 90 99 216167-95-2elsibucol
2930 90 99 168682-53-9ezatiostat
2930 90 99 58569-55-4metenkefalin
2930 90 99 887148-69-8monepantel
2930 90 99 603139-19-1odanacatib
2930 90 99 162520-00-5salirasib
2930 90 99 216167-82-7succinobucol
2930 90 99 125961-82-2tipelukast
2931 00 99 125973-56-0amsilarotene
2932 19 00 253128-41-5eribulin
2932 19 00 186953-56-0pafuramidine
2932 29 85 195883-06-8omtriptolide
2932 99 00 664338-39-0arterolane
2932 99 00 183133-96-2cabazitaxel
2932 99 00 401925-43-7celivarone
2932 99 00 461432-26-8dapagliflozin
2932 99 00 118457-15-1dexnebivolol
2932 99 00 156294-36-9larotaxel
2932 99 00 118457-16-2levonebivolol
2932 99 00 83461-56-7mifamurtide
2932 99 00 117570-53-3vadimezan
2933 19 90 496775-61-2eltrombopag
2933 19 90 206884-98-2niraxostat
2933 19 90 410528-02-8palovarotene
2933 19 90 376592-42-6totrombopag
2933 29 90 183659-72-5catramilast
2933 29 90 944263-65-4demiditraz
2933 29 90 867153-61-5dulanermin
2933 29 90 320367-13-3lixisenatide
2933 29 90 698389-00-3rolipoltide
2933 29 90 697766-75-9velafermin
2933 39 99 147084-10-4alcaftadine
2933 39 99 54-96-6amifampridine
2933 39 99 249921-19-5anamorelin
2933 39 99 319460-85-0axitinib
2933 39 99 208110-64-9befiradol
2933 39 99 330942-05-7betrixaban
2933 39 99 201034-75-5daporinad
2933 39 99 209783-80-2entinostat
2933 39 99 412950-27-7goxalapladib
2933 39 99 218791-21-0imisopasem manganese
2933 39 99 103129-82-4levamlodipine
2933 39 99 154357-42-3levonadifloxacin
2933 39 99 108147-54-2migalastat
2933 39 99 453562-69-1motesanib
2933 39 99 139145-27-0parogrelil
2933 39 99 459856-18-9pexacerfont
2933 39 99 706779-91-1pimavanserin
2933 39 99 362665-56-3pitolisant
2933 39 99 861151-12-4rosonabant
2933 39 99 701977-09-5taranabant
2933 39 99 189950-11-6tropantiol
2933 39 99 793655-64-8vapitadine
2933 39 99 139290-65-6volinaserin
2933 49 90 141388-76-3besifloxacin
2933 49 90 697761-98-1elvitegravir
2933 49 90 185055-67-8ferroquine
2933 49 90 445041-75-8intiquinatine
2933 49 90 378746-64-6nemonoxacin
2933 49 90 245765-41-7ozenoxacin
2933 49 90 412950-08-4rilapladib
2933 49 90 871224-64-5almorexant
2933 49 90 863029-99-6balamapimod
2933 49 90 698387-09-6neratinib
2933 49 90 154652-83-2tezampanel
2933 49 90 128253-31-6veliflapon
2933 59 95 791828-58-5aderbasib
2933 59 95 840486-93-3adipiplon
2933 59 95 850649-61-5alogliptin
2933 59 95 859212-16-1bafetinib
2933 59 95 380843-75-4bosutinib
2933 59 95 839712-12-8cariprazine
2933 59 95 414910-27-3casopitant
2933 59 95 288383-20-0cediranib
2933 59 95 849550-05-6cevipabulin
2933 59 95 827318-97-8danusertib
2933 59 95 356057-34-6darapladib
2933 59 95 501000-36-8dutacatib
2933 59 95 247257-48-3fimasartan
2933 59 95 3432-99-3folitixorin
2933 59 95 668270-12-0linagliptin
2933 59 95 441798-33-0macitentan
2933 59 95 641571-10-0nilotinib
2933 59 95 763113-22-0olaparib
2933 59 95 686344-29-6otenabant
2933 59 95 625115-55-1riociguat
2933 59 95 486460-32-6sitagliptin
2933 59 95 425637-18-9sotrastaurin
2933 59 95 309913-83-5talmapimod
2933 59 95 113857-87-7talotrexin
2933 59 95 274693-27-5ticagrelor
2933 59 95 306296-47-9vicriviroc
2933 69 80 775351-65-0imeglimin
2933 79 00 461443-59-4aplaviroc
2933 79 00 189691-06-3bremelanotide
2933 79 00 813452-18-5carmegliptin
2933 79 00 405169-16-6dovitinib
2933 79 00 536748-46-6eribaxaban
2933 79 00 473289-62-2ilepatril
2933 79 00 180694-97-7mimopezil
2933 79 00 579475-18-6orvepitant
2933 79 00 449811-01-2pamapimod
2933 79 00 248282-01-1paquinimod
2933 79 00 380917-97-5perampanel
2933 79 00 552292-08-7rolapitant
2933 79 00 425386-60-3semagacestat
2933 79 00 515814-01-4voclosporin
2933 99 80 481629-87-2aleplasinin
2933 99 80 394730-60-0boceprevir
2933 99 80 649735-63-7brivanib alaninate
2933 99 80 483369-58-0denagliptin
2933 99 80 284019-34-7denibulin
2933 99 80 481631-45-2diaplasinin
2933 99 80 272105-42-7disitertide
2933 99 80 227318-71-0epetirimod
2933 99 80 259793-96-9favipiravir
2933 99 80 871576-03-3flovagatran
2933 99 80 229305-39-9golotimod
2933 99 80 258818-34-7larazotide
2933 99 80 571170-77-9laropiprant
2933 99 80 616202-92-7lorcaserin
2933 99 80 868771-57-7melogliptin
2933 99 80 803712-67-6obatoclax
2933 99 80 404950-80-7panobinostat
2933 99 80 625114-41-2piragliatin
2933 99 80 74847-35-1pyronaridine
2933 99 80 872178-65-9rabeximod
2933 99 80 355151-12-1rotigaptide
2933 99 80 497221-38-2rusalatide
2933 99 80 187602-11-5sofigatran
2933 99 80 227318-75-4sotirimod
2933 99 80 402957-28-2telaprevir
2933 99 80 848084-83-3tigapotide
2933 99 80 393105-53-8tiplasinin
2933 99 80 620948-93-8vabicaserin
2933 99 80 794466-70-9vernakalant
2934 10 00 544417-40-5capadenoson
2934 10 00 302962-49-8dasatinib
2934 10 00 223132-37-4inolitazone
2934 10 00 241479-67-4isavuconazole
2934 10 00 338990-84-4isavuconazonium chloride
2934 10 00 607723-33-1lobeglitazone
2934 10 00 280782-97-0managlinat dialanetil
2934 10 00 790299-79-5masitinib
2934 10 00 223673-61-8mirabegron
2934 10 00 501948-05-6rosabulin
2934 10 00 447406-78-2sodelglitazar
2934 10 00 760937-92-6teneligliptin
2934 20 80 848344-36-5bentamapimod
2934 20 80 870093-23-5talarozole
2934 99 90 320345-99-1aclidinium bromide
2934 99 90 222551-17-9adoprazine
2934 99 90 207623-20-9agatolimod
2934 99 90 475479-34-6aleglitazar
2934 99 90 870524-46-2amolimogene bepiplasmid
2934 99 90 875446-37-0anacetrapib
2934 99 90 250386-15-3apadenoson
2934 99 90 541550-19-0apilimod
2934 99 90 160707-69-7apricitabine
2934 99 90 147403-03-0azilsartan
2934 99 90 863031-21-4azilsartan medoxomil
2934 99 90 757942-43-1bederocin
2934 99 90 627861-07-8beperminogene perplasmid
2934 99 90 959961-96-7bevasiranib
2934 99 90 769901-96-4capeserod
2934 99 90 868540-17-4carfilzomib
2934 99 90 872847-66-0cenersen
2934 99 90 80295-38-1conestat alfa
2934 99 90 903916-27-8custirsen
2934 99 90 187865-22-1derquantel
2934 99 90 134379-77-4dexelvucitabine
2934 99 90 247046-52-2dilopetine
2934 99 90 480449-70-5edoxaban
2934 99 90 188181-42-2elacytarabine
2934 99 90 98819-76-2esreboxetine
2934 99 90 763903-67-9fosalvudine tidoxil
2934 99 90 172673-20-0fosaprepitant
2934 99 90 522664-63-7ibodutant
2934 99 90 405159-59-3idrabiotaparinux sodium
2934 99 90 188116-07-6imepitoin
2934 99 90 335619-18-6inakalant
2934 99 90 1391-36-2lancovutide
2934 99 90 189059-71-0lapaquistat
2934 99 90 327026-93-7lensiprazine
2934 99 90 170632-47-0lificiguat
2934 99 90 852313-25-8litenimod
2934 99 90 1000120-98-8mipomersen
2934 99 90 62253-63-8nepidermin
2934 99 90 26833-87-4omacetaxine mepesuccinate
2934 99 90 269718-84-5pardoprunox
2934 99 90 219923-85-0pramiconazole
2934 99 90 377727-87-2preladenant
2934 99 90 524684-52-4prinaberel
2934 99 90 865311-47-3quarfloxin
2934 99 90 869884-78-6radezolid
2934 99 90 496054-87-6radiprodil
2934 99 90 518048-05-0raltegravir
2934 99 90 787548-03-2regrelor
2934 99 90 820957-38-8retosiban
2934 99 90 572924-54-0ridaforolimus
2934 99 90 128517-07-7romidepsin
2934 99 90 93265-81-7ropidoxuridine
2934 99 90 151823-14-2sapacitabine
2934 99 90 379231-04-6saracatinib
2934 99 90 791635-59-1simotaxel
2934 99 90 119567-79-2taribavirin
2934 99 90 332012-40-5telatinib
2934 99 90 925681-61-4trabedersen
2934 99 90 189003-92-7trelanserin
2934 99 90 296251-72-4velimogene aliplasmid
2934 99 90 904302-98-3viquidacin
2934 99 90 872525-61-6votucalis
2934 99 90 221877-54-9zotarolimus
2935 00 90 197904-84-0apricoxib
2935 00 90 769169-27-9begacestat
2935 00 90 414864-00-9belinostat
2935 00 90 313682-08-5brecanavir
2935 00 90 839673-52-8cevoglitazar
2935 00 90 358970-97-5drinabant
2935 00 90 865200-20-0giripladib
2935 00 90 464213-10-3ibipinabant
2935 00 90 173424-77-6laromustine
2935 00 90 398507-55-6lodenafil carbonate
2935 00 90 136564-68-6masilukast
2935 00 90 170569-88-7mavacoxib
2935 00 90 862189-95-5mirodenafil
2935 00 90 439687-69-1nelivaptan
2935 00 90 691852-58-1nesbuvir
2935 00 90 778576-62-8oglemilast
2935 00 90 444731-52-6pazopanib
2935 00 90 362505-84-8relacatib
2935 00 90 243984-11-4resatorvid
2935 00 90 519055-62-0tasisulam
2935 00 90 186497-07-4zibotentan
2936 29 00 104121-92-8eldecalcitol
2936 29 00 31690-09-2levomefolic acid
2937 19 00 782500-75-8albiglutide
2937 19 00 348119-84-6obinepitide
2937 19 00 295350-45-7ozarelix
2937 19 00 275371-94-3taspoglutide
2937 19 00 218949-48-5tesamorelin
2937 19 00 22006-64-0tridecactide
2937 22 00 132245-57-9dexamethasone cipecilate
2937 22 00 397864-44-7fluticasone furoate
2937 29 00 211254-73-8lonaprisan
2937 50 00 333963-42-1cobiprostone
2937 50 00 172740-14-6posaraprost
2937 90 00 834153-87-6elagolix
2937 90 00 609799-22-6tasimelteon
2937 90 00 342577-38-2velneperit
2939 19 00 73232-52-7methylnaltrexone bromide
2939 59 00 136199-02-5rolofylline
2939 99 00 850607-58-8darotropium bromide
2939 99 00 187852-63-7delimotecan
2940 00 00 9007-72-1ferric carboxymaltose
2940 00 00 442201-24-3remogliflozin etabonate
2940 00 00 408504-26-7sergliflozin etabonate
2941 90 00 467214-20-6alvespimycin
2941 90 00 677017-23-1berubicin
2941 90 00 229016-73-3ceftaroline fosamil
2941 90 00 318498-76-9flopristin
2941 90 00 145435-72-9gamithromycin
2941 90 00 325965-23-9linopristin
2941 90 00 857402-23-4retaspimycin
2941 90 00 305841-29-6sagopilone
2941 90 00 75747-14-7tanespimycin
2941 90 00 328898-40-4tildipirosin
2941 90 00 222400-20-6tomopenem
2941 90 00 63409-12-1tylvalosin
3001 90 91 9041-08-1semuloparin sodium
3002 10 91 792921-10-9abagovomab
3002 10 91 910649-32-0anrukinzumab
3002 10 91 648904-28-3bavituximab
3002 10 91

402710-27-4

(light chain)

402710-25-2

(heavy chain)

canakinumab
3002 10 99 945228-49-9citatuzumab bogatox
3002 10 91 880486-59-9dacetuzumab
3002 10 91 615258-40-7denosumab
3002 10 91 762260-74-2efungumab
3002 10 91 89957-37-9gantenerumab
3002 10 91 680188-33-4ibalizumab
3002 10 91 477202-00-9ipilimumab
3002 10 91 640735-09-7iratumumab
3002 10 91 845816-02-6lexatumumab
3002 10 91 903512-50-5lucatumumab
3002 10 91 899796-83-9milatuzumab
3002 10 91 677010-34-3motavizumab
3002 10 91 676258-98-3naptumomab estafenatox
3002 10 91 828933-51-3nimotuzumab
3002 10 91 949142-50-1obinutuzumab
3002 10 91 637334-45-3ocrelizumab
3002 10 91 881191-44-2otelixizumab
3002 10 91 372075-37-1sontuzumab
3002 10 91 705287-60-1stamulumab
3002 10 91 339086-80-5tadocizumab
3002 10 91

592557-43-2

(light chain)

592557-41-0

(heavy chain)

tenatumomab
3002 10 91 876387-05-2teplizumab
3002 10 91 918127-53-4tigatuzumab
3002 10 91 745013-59-6tremelimumab
3002 10 91 339986-90-2tucotuzumab celmoleukin
3002 10 91 728917-18-8veltuzumab
3002 10 91 896731-82-1conatumumab
3002 10 91 892553-42-3etaracizumab
3002 10 91 944548-38-3foravirumab
3002 10 91 944548-37-2rafivirumab
3002 10 91 880266-57-9tanezumab
3002 10 91 815610-63-0ustekinumab
3002 10 95 862111-32-8aflibercept
3002 10 95 845264-92-8atacicept
3002 10 95 909110-25-4baminercept
3002 10 95 9001-27-8beroctocog alfa
3002 10 95 879555-13-2epoetin kappa
3002 10 95 762263-14-9epoetin theta
3002 10 95 501081-76-1rilonacept
3002 10 95 267639-76-9romiplostim
3002 10 95 869858-13-9thrombin alfa
3002 10 95 897936-89-9vatreptacog alfa (activated)
3002 10 95 472960-22-8albinterferon alfa-2b
3002 10 95 869881-54-9briobacept
3002 10 95 606138-08-3catridecacog
3002 10 95 716840-32-3denenicokin
3002 10 95 931101-84-7troplasminogen alfa
3002 10 99 934216-54-3alacizumab pegol
3002 20 00 181477-43-0disomotide
3002 20 00 181477-91-8ovemotide
3002 20 00 915019-08-8tertomotide
3002 20 00 295371-00-5verpasep caltespen
3002 90 90 473553-86-5alferminogene tadenovec
3002 90 90 929881-05-0alipogene tiparvovec
3002 90 90 600735-73-7contusugene ladenovec
3002 90 90 851199-59-2linaclotide
3002 90 90 898830-54-1sitimagene ceradenovec
3002 90 90 721946-42-5transferrin aldifitox
3507 90 90 9026-00-0bucelipase alfa
3507 90 90 885051-90-1pegloticase
3507 90 90 884604-91-5velaglucerase alfa
3911 90 99 892497-01-7azoximer bromide

Annex IIList of prefixes and suffixes which, in combination with the INNs of Annex 3 to Annex I to Regulation (EEC) No 2658/87, describe the salts, esters or hydrates of INNs; these salts, esters and hydrates are free of duty, on condition that they are classifiable in the same six-digit HS subheading as the corresponding INN

The references to ‘International Nonproprietary Names (INN) for pharmaceutical substances, names for radicals and groups, comprehensive list 2004’ are replaced by ‘International Nonproprietary Names (INN) for pharmaceutical substances, names for radicals, groups and others, comprehensive list 2007’.

The following prefixes or suffixes are added to the list included in Annex 4 to Annex I to Regulation (EEC) No 2658/87:

Preferred prefix or suffixSynonymSystematic name when different
alanetil (INNRG) [(S)-1-ethoxy-1-oxo-propan-2-yl]amino (INNCN)
alaninate (INNRG) L-alaninate (INNCN)
alapivoxil (INNRG) L-alanyl, [(2,2-dimethylpropanoyl)oxy]metyl (INNCN)
aldifitox (INNRG) (4-iminobutane-1,4-diyl)sulfanediyl[(3RS)-2,5-dioxopyrrolidine-1,3-diyl]-1,3-phenylenecarbonyl and forming an N-benzoyl derivative of a primary amine group of diphtheria [550-L-phenylalanine]toxin from Corynebacterium diphtheriae-(26-560)-peptide (INNCN)
besudotox (INNRG) L-lysyl-L-alanyl-L-serylglycylglycine (linker) fusion protein with des-(365-380)-[Asn364,Val407,Ser515,Gln590,Gln606,Arg613]exotoxin A (Pseudomonas aeruginosa)-(251-613)-peptide (toxin with region IA and first 16 residues of region IB deleted) (INNCN)
ceribate (INNRG) rac-2,3-dihydroxypropyl carbonate (ester) (INNCN)
cipecilate (INNRG) cyclohexanecarboxylate (ester), cyclopropanecarboxylate (ester) (INNCN)
dalanated (INNRG) des-B30-alanine (INNCN)
enacarbil (INNRG) {rac-1-[(2-methylpropanoyl)oxy]ethoxy}carbonyl (INNCN)
estafenatox (INNRG) glycylglycyl-L-proline (linker) fusion protein with enterotoxin type A (Staphylococcus aureus)-(1-33)-peptidyl-L-seryl[Ser36,Ser37,Glu38,Lys39,Ala41,Thr46,Thr71,Ala72,Ser75,Glu76,Glu78,Ser80,Ser81,Thr214,Ser217,Thr219,Ser220,Ser222,Ser224]enterotoxin type E (Staphylococcus aureus)-(32-230)-peptide (synthetic superantigen SEA/E-120) (INNCN)
etexilate (INNRG) ethyl, (hexyloxy)carbonyl
fosamil (INNRG) phosphono (INNCN)
glucuronide (INNRG) β-D-glucopyranosiduronic acid [oside] (INNCN)
medocaril (INNRG) [(5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy]carbonyl (INNCN)
paptox (INNRG) protein PAP (Phytolacca americana antiviral) (INNCN)
placarbil (INNRG) (R)-2-methyl-1-[(2-methylpropanoyl)oxy]propoxy}carbonyl) (INNCN)

The systematic name of the following prefix or suffix is amended as follows:

Preferred prefix or suffixSynonymSystematic name when different
aritox (INNRG) ricin A chain (INNCN)

Annex III

List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be added to the list of products receiving duty-free treatment included in Annex 6 to Annex I to Regulation (EEC) No 2658/87

CN codeCAS RNName
2843 29 00 22199-08-2[4-amino-N-(pyrimidin-2(1H)-ylidene-κN1)benzenesulfonamidato-κO]silver
2905 39 95 281214-27-5(2R,3R)-2,3-dimethylbutane-1,4-diyl bis(4-methylbenzenesulfonate)
2905 59 98 441002-17-14-chlorobutyl 2-nitrobenzenesulfonate
2909 30 90 92878-95-02-(3-chloropropoxy)-1-methoxy-4-nitrobenzene
2909 30 503070-57-32-({2-[(6-bromohexyl)oxy]ethoxy}methyl)-1,3-dichlorobenzene
2909 30 461432-23-54-(5-bromo-2-chlorobenzyl)phenyl ethyl ether
2909 49 80 185954-75-0(3R)-3-methoxydecan-1-ol
2909 49 80 85309-91-72-[(2,6-dichlorobenzyl)oxy]ethanol
2909 49 80 160969-03-92-[2-(2,2,2-trifluoroethoxy)phenoxy]ethyl methanesulfonate
2909 50 00 167145-13-32-[2-(3-methoxyphenyl)ethyl]phenol
2910 20 00 15448-47-2(2R)-2-methyloxirane
2910 90 00 62600-71-9(2R)-2-(3-chlorophenyl)oxirane
2910 90 00 702687-42-1(2R)-2-[(5-bromo-2,3-difluorophenoxy)methyl]oxirane
2910 90 00 683276-64-4[(2R)-2-methyloxiran-2-yl]methyl 4-nitrobenzenesulfonate
2913 00 00 90035-34-04′-(trifluoromethyl)biphenyl-4-carbaldehyde
2914 40 90 17752-16-8(3β)-3-hydroxycholest-5-en-24-one
2914 50 00 974-23-2(3β,16α)-3-hydroxy-16,17-epoxypregn-5-en-20-one
2914 70 00 13054-81-44-chloro-heptane-3,5-dione
2914 70 00 10226-30-96-chlorohexan-2-one
2915 60 90 53064-79-2iodomethyl pivalate
2915 90 00 22328-90-1(3R)-3-methylhexanoic acid
2915 90 00 1069-66-5sodium 2-propylpentanoate
2916 20 00 211515-46-71-(2-ethylbutyl)cyclohexanecarbonyl chloride
2916 20 00 381209-09-21-(2-ethylbutyl)cyclohexanecarboxylic acid
2916 20 00 7077-05-6trans-4-(propan-2-yl)cyclohexanecarboxylic acid
2916 39 00 21900-39-05-fluoro-2-methylbenzoyl chloride
2916 39 00 17625-03-5sodium hydrogen 3-sulfonatobenzoate
2917 19 90 76-72-2diethyl ethyl(pentan-2-yl)propanedioate
2918 29 00 376592-58-45′-chloro-2′-hydroxy-3′-nitrobiphenyl-3-carboxylic acid
2918 99 90 709031-28-7(3-hydroxytricyclo[3.3.1.1(3,7)]dec-1-yl)(oxo)acetic acid
2918 99 90 35480-52-52,5-bis(2,2,2-trifluoroethoxy)benzoic acid
2918 99 90 4651-67-6(3α,5β)-3-hydroxy-7-oxocholan-24-oic acid
2918 99 90 52179-28-9ethyl 2-[4-(2,2-dichlorocyclopropyl)phenoxy]-2-methylpropanoate
2918 99 90 530141-60-7methyl 3-(5-{[4-(cyclopentyloxy)-2-hydroxyphenyl]carbonyl}-2-hydroxyphenyl)propanoate
2920 90 10 91526-18-04-(hydroxymethyl)-5-methyl-1,3-dioxol-2-one
2921 49 00 334477-60-0(1R)-1-[3,5-bis(trifluoromethyl)phenyl]-N-methylethanamine
2921 49 00 376608-71-8(1R,2S)-2-(3,4-difluorophenyl)cyclopropanaminium (2R)-hydroxy(phenyl)ethanoate
2921 49 00 1034457-07-22-(2,3-dihydro-1H-inden-2-yl)propan-2-amine hydrochloride
2921 49 00 945717-05-52-(4-chloro-3-ethylphenyl)ethanamine hydrochloride
2921 49 00 89-97-42-chlorobenzylamine
2921 49 00 945717-43-1N-(4-tert-butylbenzyl)-2-(4-chloro-3-ethylphenyl)ethanamine
2921 51 90 150812-21-8N4-[(4-fluorophenyl)methyl]-2-nitro-1,4-benzenediamine
2922 19 85 1035455-90-3(2R)-1-(5-bromo-2,3-difluorophenoxy)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}propan-2-ol hydrochloride
2922 19 85 0-00-0[2-(chloromethyl)-4-(dibenzylamino)phenyl]methanol hydrochloride
2922 19 85 133-51-7antimonic acid – 1-deoxy-1-(methylamino)-D-glucitol (1:1)
2922 19 85 1035455-87-8ethyl (2E)-3-(3-{[(2R)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}-2-hydroxypropyl]oxy}-4,5-difluorophenyl)prop-2-enoate hydrochloride
2922 19 85 702686-97-3ethyl 3-(3-{[(2R)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}-2-hydroxypropyl]oxy}-4,5-difluorophenyl)propanoate hydrochloride
2922 29 00 20059-73-82-[4-(aminomethyl)phenoxy]-N,N-dimethylethanamine
2922 49 85 848133-35-7(2E)-4-(dimethylamino)but-2-enoic acid hydrochloride
2922 49 85 610300-07-7(3S,5R)-3-amino-5-methyloctanoic acid
2922 49 85 610300-00-0(3S,5R)-3-amino-5-methyloctanoic acid hydrochloride
2922 49 85 143785-86-84-(1-aminocyclopropyl)-2,3,5-trifluorobenzoic acid
2922 49 85 848949-85-94-fluoro-L-leucine – ethyl hydrogen sulfate (1:1)
2922 49 85 39068-93-4methyl 2-(dimethylamino)-2-phenylbutanoate
2922 49 85 168619-25-8methyl 3′-aminobiphenyl-3-carboxylate
2922 49 85 82834-12-6N-[(2S)-1-ethoxy-1-oxopentan-2-yl]-L-alanine
2922 49 85 94133-84-3sodium 2-amino-2-phenylbutanoate
2922 50 00 503070-58-4triphenylacetic acid – 4-{(1R)-2-[(6-{2-[(2,6-dichlorobenzyl)oxy]ethoxy}hexyl)amino]-1-hydroxyethyl}-2-(hydroxymethyl)phenol (1:1)
2924 19 00 62009-47-62-aminomalonamide
2924 19 00 7355-58-0N-(2-chloroethyl)acetamide
2924 29 98 361442-00-4{2-[(tert-butoxycarbonyl)amino]-3-hydroxytricyclo[3.3.1.1(3,7)]dec-1-yl}acetic acid
2924 29 98 266993-72-02,3-diaminobenzamide dihydrochloride
2924 29 98 168080-49-72-chloro-4-{[(5-fluoro-2-methylphenyl)carbonyl]amino}benzoic acid
2924 29 98 317374-08-62-methyl-4-{[(2-methylphenyl)carbonyl]amino}benzoic acid
2924 29 98 143785-84-64-(1-carbamoylcyclopropyl)-2,3,5-trifluorobenzoic acid
2924 29 98 143785-87-94-[1-(acetylamino)cyclopropyl]-2,3,5-trifluorobenzoic acid
2924 29 98 108166-22-94-{[(2-methylphenyl)carbonyl]amino}benzoic acid
2924 29 98 150812-23-0ethyl {4-[(4-fluorobenzyl)amino]-2-nitrophenyl}carbamate
2924 29 98 22316-45-6ethyl 3-[(5-chloro-2-nitrophenyl)(phenyl)amino]-3-oxopropanoate
2924 29 98 316173-29-2methyl (1S,2S,3S,4R)-3-[(1S)-1-amino-2-ethylbutyl]-4-[(tert-butoxycarbonyl)amino]-2-hydroxycyclopentanecarboxylate
2924 29 98 1142-20-7N-benzyloxycarbonyl-L-alanine
2924 29 98 84996-93-0N-cyclohexyl-5-hydroxypentanamide
2924 29 98 579494-66-9propyl {4-[2-(diethylamino)-2-oxoethoxy]-3-ethoxyphenyl}acetate
2925 19 95 265136-65-0ethyl 3-amino-4-[2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)ethoxy]but-2-enoate
2926 90 95 855425-38-61-(2-ethylbutyl)cyclohexanecarbonitrile
2926 90 95 846023-24-32-cyano-N-(2,4-dichloro-5-methoxyphenyl)acetamide
2926 90 95 591769-05-03-cyclopentylprop-2-enenitrile
2926 90 95 20099-89-24-(bromoacetyl)benzonitrile
2926 90 95 474554-45-54,5-diethoxy-3-fluorobenzene-1,2-dicarbonitrile
2926 90 95 79370-78-85-hydroxybenzene-1,3-dicarbonitrile
2926 90 95 139481-28-0methyl 2-{[(2′-cyanobiphenyl-4-yl)methyl]amino}-3-nitrobenzoate
2928 00 90 860035-10-51-({[(2,5-dioxopyrrolidin-1-yl)oxy]carbonyl}oxy)ethyl 2-methylpropanoate
2928 00 90 910656-45-02-hydroxy-2-(trifluoromethyl)butanehydrazide
2928 00 90 95759-10-74-chloro-2-[(2-methoxy-2-oxoethoxy)imino]-3-oxobutanoic acid
2928 00 90 473927-63-8ethyl (2Z)-chloro[2-(4-methoxyphenyl)hydrazinylidene]ethanoate
2928 00 90 158671-29-5N,2-dihydroxy-4-methylbenzamide
2928 00 90 84080-68-2tert-butyl (2Z)-2-[(2-methoxy-2-oxoethoxy)imino]-3-oxobutanoate
2928 00 90 268544-50-9tert-butyl-2-[(2-methoxy-2-oxoethoxy)imino]-3-oxobutanoate
2930 90 99 13459-62-6{2-[(4-chlorophenyl)sulfanyl]phenyl}acetic acid
2930 90 99 211513-21-21-(2-ethylbutyl)-N-(2-sulfanylphenyl)cyclohexanecarboxamide
2930 90 99 860035-07-01-{[(methylsulfanyl)carbonyl]oxy}ethyl 2-methylpropanoate
2930 90 99 893407-18-62,2,2-trifluoro-1-[4′-(methylsulfonyl)biphenyl-4-yl]ethanone
2930 90 99 60759-00-43,4-diethoxybenzenecarbothioamide
2930 90 99 21048-05-5N-methylbenzenecarbothiohydrazide
2931 00 99 13682-94-5(2-bromoethenyl)(trimethyl)silane
2931 00 99 914922-89-7(2R,4R)-4-[[(1,1-dimethylethyl)dimethylsilyl]oxy]-N-methoxy-N,2-dimethyl-7-oxoheptanamide
2931 00 99 914922-88-6(2R,4R)-4-{[tert-butyl(dimethyl)silyl]oxy}-N-methoxy-N,2-dimethyloct-7-enamide
2931 00 99 871355-80-5(4R)-2-bromo-7-{[tert-butyl(diphenyl)silyl]oxy}hept-1-en-4-yl 4-methylbenzenesulfonate
2931 00 99 89694-48-4(5-chloro-2-methoxyphenyl)boronic acid
2931 00 99 701278-08-2[(1R,5S)-5-[dimethyl(phenyl)silyl]-2-{[(2-methoxypropan-2-yl)oxy]methyl}cyclopent-2-en-1-yl]methanol
2931 00 99 701278-09-3{(4S,5R)-5-[(benzyloxy)methyl]-4-[dimethyl(phenyl)silyl]cyclopent-1-en-1-yl}methanol
2931 00 99 796967-18-51-(2-fluoro-5-methylphenyl)-3-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]urea
2931 00 99 172732-52-42-(1,3,2-dioxaborinan-2-yl)benzonitrile
2931 00 99 185411-12-5methyl 3-(trimethylsilyl)pent-4-enoate
2932 19 00 253128-10-8(1S)-1,5:7,10-dianhydro-12,13-bis-O-[tert-butyl(dimethyl)silyl]-2,3,4,6,8,11-hexadeoxy-1-{2-[(2S,5S)-5-(3-hydroxypropyl)-3-methylidenetetrahydrofuran-2-yl]ethyl}-3-methyl-9-O-methyl-4-methylidene-8-[(phenylsulfonyl)methyl]-D-arabino-D-altro-tridecitol
2932 19 00 441045-17-6(1S,3S,6S,9S,12S,14R,16R,18S,20R,21R,22S,26R,29S,31R,32S,33R,35R,36S)-20-[(2S)-3-amino-2-hydroxypropyl]-21-methoxy-14-methyl-8,15-bis(methylene)-2,19,30,34,37,39,40,41-octaoxanonacyclo[24.9.2.13,32.13,33.16,9.112,16.018,22.029,36.031,35]hentetracontan-24-one methanesulfonate
2932 29 85 916069-80-2(4S)-4-(fluoromethyl)dihydrofuran-2(3H)-one
2932 29 85 63106-93-41-phenyl-3-oxabicyclo[3.1.0]hexan-2-one
2932 29 85 7734-80-72-oxo-2H-chromene-6-carboxylic acid
2932 29 85 0-00-04-(4-fluorophenyl)-7-(isothiocyanatomethyl)-2H-chromen-2-one
2932 29 85 947408-91-56-[(2,4-dihydroxyphenyl)carbonyl]-2H-chromen-2-one
2932 29 85 947408-90-46-[(2,4-dimethoxyphenyl)carbonyl]-2H-chromen-2-one
2932 99 00 452342-08-4(1R)-2-(benzylamino)-1-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)ethanol
2932 99 00 99541-23-8(1R,2S,3R,4R,5R)-4-azido-2-{[(4aR,6S,7R,8S,8aR)-7,8-bis(benzyloxy)-2-phenylhexahydropyrano[3,2-d][1,3]dioxin-6-yl]oxy}-6,8-dioxabicyclo[3.2.1]oct-3-yl acetate
2932 99 00 461432-25-7(1S)-2,3,4,6-tetra-O-acetyl-1,5-anhydro-1-[4-chloro-3-(4-ethoxybenzyl)phenyl]-D-glucitol
2932 99 00 196597-79-2(2E)-1,2,6,7-tetrahydro-8H-indeno[5,4-b]furan-8-ylideneethanenitrile
2932 99 00 3308-94-92-(3-chloropropyl)-2-(4-fluorophenyl)-1,3-dioxolane
2932 99 00 274693-53-7[(3aS,4R,6S,6aR)-6-hydroxy-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl]carbamate
2932 99 00 185954-98-7[6(2Z,3R)]-3-O-decyl-2-deoxy-6-O-[2-deoxy-3-O-(3-metoxydecyl)-6-methyl-2-[(1-oxo-11-octadecenyl)amino]-4-O-phosphono-β-D-glucopyranosyl]-2-[(1,3-dioxotetradecyl)amino]-α-D-glucopyranose 1-(dihydrogen phosphate) tetrasodium salt
2932 99 00 136172-58-21,6-di-O-acetyl-2-azido-3,4-di-O-benzyl-2-deoxy-D-glucopyranose
2932 99 00 196597-80-52-[(8S)-1,6,7,8-tetrahydro-2H-indeno[5,4-b]furan-8-yl]ethanamine hydrochloride
2932 99 00 666860-59-92-amino-2-oxoethyl{3-[trans-5-(6-methoxynaphthalen-1-yl)-1,3-dioxan-2-yl]propyl}carbamate
2932 99 00 117661-72-05-(chloromethyl)-6-methyl-1,3-benzodioxole
2932 99 00 959624-24-96-(hydroxymethyl)-4-phenyl-3,4-dihydro-2H-chromen-2-ol
2932 99 00 960404-59-5but-2-yne-1,4-diol – methyl 1-C-[4-chloro-3-(4-ethoxybenzyl)phenyl]-α-D-glucopyranoside (1:1)
2932 99 00 15826-37-6disodium 5,5′-[(2-hydroxypropane-1,3-diyl)bis(oxy)]bis(4-oxo-4H-chromene-2-carboxylate)
2932 99 00 204254-84-2ethyl (3aR,7R,7aR)-2,2-dimethyl-7-[(methylsulfonyl)oxy]-3a,6,7,7a-tetrahydro-1,3-benzodioxole-5-carboxylate
2932 99 00 99541-26-1methyl (2S,3S,4S,5S,6S)-6-{[(1S,2S,3S,4R,5R)-3-(acetyloxy)-4-azido-6,8-dioxabicyclo[3.2.1]oct-2-yl]methyl}-4,5-bis(benzyloxy)-3-hydroxytetrahydro-2H-pyran-2-carboxylate
2932 99 00 114869-97-5methyl 6-O-acetyl-4-O-(2-O-acetyl-3-O-benzyl-6-methyl-α-L-idopyranuronosyl)-3-O-benzyl-2-{[(benzyloxy)carbonyl]amino}-2-deoxy-α-D-glucopyranoside
2933 19 90 1035677-60-1(4S)-3-(4-chlorophenyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide 2,3-dihydroxybutanedioate
2933 19 90 18048-64-12-(3,4-dimethylphenyl)-5-methyl-2,4-dihydro-3H-pyrazol-3-one
2933 19 90 1035675-24-13-(4-chlorophenyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide
2933 19 90 1028026-83-65-methyl-1-(propan-2-yl)-4-[4-(propan-2-yloxy)benzyl]-1,2-dihydro-3H-pyrazol-3-one
2933 19 90 473921-12-95-{[3,5-diethyl-1-(2-hydroxyethyl)-1H-pyrazol-4-yl]oxy}benzene-1,3-dicarbonitrile
2933 29 90 65902-59-22-bromo-4-nitro-1H-imidazole
2933 29 90 57531-37-02-chloro-4-nitro-1H-imidazole
2933 29 90 1000164-35-13-(1,1-dimethylethyl)-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-1-(triphenylmethyl)-L-histidyl-2-methylalanyl-L-α-glutamylglycine
2933 29 90 152074-97-0L-α-aspartyl-L-α-glutamyl-L-asparaginyl-L-prolyl-L-valyl-L-valyl-L-histidyl-L-phenylalanyl-L-phenylalanyl-L-lysyl-L-asparaginyl-L-isoleucyl-L-valyl-L-threonyl-L-prolyl-L-arginyl-L-threonine
2933 29 90 781666-30-6L-α-aspartyl-L-α-glutamyl-L-asparaginyl-L-prolyl-L-valyl-L-valyl-L-histidyl-L-phenylalanyl-L-phenylalanyl-L-lysyl-L-asparaginyl-L-isoleucyl-L-valyl-L-threonyl-L-prolyl-L-arginyl-L-threonine tetraacetate
2933 29 90 451470-33-0methyl 3′-(2-methyl-4,5-dihydro-1H-imidazol-1-yl)biphenyl-3-carboxylate
2933 39 99 925978-49-0(+)-5-[6-(1-methyl-1H-pyrazol-4-yl)pyridin-3-yl]-1-azabicyclo[3.2.1]octane
2933 39 99 876170-44-4(1S,5S)-3-(5,6-dichloropyridin-3-yl)-3,6-diazabicyclo[3.2.0]heptane benzenesulfonate
2933 39 99 741705-70-4(2R)-phenyl[(2R)-piperidin-2-yl]ethanoic acid hydrochloride
2933 39 99 414910-13-7(2S)-hydroxy(phenyl)ethanoic acid – (2R)-2-(4-fluoro-2-methylphenyl)piperidin-4-one (1:1)
2933 39 99 0-00-0(3aR,6aR)-1-(pyridin-3-yl)octahydropyrrolo[3,4-b]pyrrole 4-methylbenzenesulfonate
2933 39 99 370882-57-8(3aR,6aR)-1-(pyridin-3-yl)octahydropyrrolo[3,4-b]pyrrole dihydrochloride
2933 39 99 334618-23-4(3R)-piperidin-3-amine dihydrochloride
2933 39 99 1062580-52-2(3R,4R)-1-benzyl-N,4-dimethylpiperidin-3-amine dihydrochloride
2933 39 99 27262-47-1(S)-1-butyl-N-(2,6-dimethylphenyl)piperidine-2-carboxamide
2933 39 99 105812-81-5[(3S,4R)-4-(4-fluorophenyl)-1-methylpiperidin-3-yl]methanol
2933 39 99 876068-51-8[(3S,4S)-4-amino-1-(5,6-dichloropyridin-3-yl)pyrrolidin-3-yl]methanol
2933 39 99 871022-14-91-({4-[({[2-oxo-3-(propan-2-yl)-2,3-dihydro-1H-benzimidazol-1-yl]carbonyl}amino)methyl]piperidin-1-yl}methyl)cyclobutanecarboxylic acid
2933 39 99 5421-92-11-(pyridin-4-yl)pyridinium chloride hydrochloride
2933 39 99 272776-12-21,1′-binaphthalene-2,2′-diol –5-methoxy-2-{(S)-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]sulfinyl}-1H-benzimidazole (1:1)
2933 39 99 871022-19-41-[(4-{[(tert-butoxycarbonyl)amino]methyl}piperidin-1-yl)methyl]cyclobutanecarboxylic acid
2933 39 99 3613-73-82,8-dimethyl-5-[2-(6-methylpyridin-3-yl)ethyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
2933 39 99 179687-79-72-[(2-chloro-4-nitrophenoxy)methyl]pyridine
2933 39 99 122321-04-42-[methyl(pyridin-2-yl)amino]ethanol
2933 39 99 945405-37-82-methyl-3-[(2S)-pyrrolidin-2-ylmethoxy]pyridine 2,3-dihydroxybutanedioate
2933 39 99 936637-40-03,3′-piperidine-1,4-diyldipropan-1-ol 4-methylbenzenesulfonate
2933 39 99 88150-62-33-ethyl-5-methyl-4-(2-chlorophenyl)-2-{[2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)ethoxy]methyl}-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate
2933 39 99 84100-54-94-(ethylamino)piperidine-4-carboxamide
2933 39 99 873546-30-64,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]bis(N′-hydroxybenzenecarboximidamide)
2933 39 99 873546-74-84,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]bis[N′-(acetyloxy)benzenecarboximidamide]
2933 39 99 873546-38-44,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]dibenzenecarboximidamide trihydrochloride pentahydrate
2933 39 99 873546-80-64,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]dibenzonitrile
2933 39 99 78750-61-54-[(3-nitropyridin-2-yl)amino]phenol
2933 39 99 866109-93-54-{4-[4-(trifluoromethoxy)phenoxy]piperidin-1-yl}phenol 4-methylbenzenesulfonate
2933 39 99 927889-51-84-bromo-2,6-diethylpyridine 4-methylbenzenesulfonate
2933 39 99 691882-47-04-hydroxybenzoic acid – (2S,4E)-N-methyl-5-[5-(propan-2-yloxy)pyridin-3-yl]pent-4-en-2-amine (1:1)
2933 39 99 876068-46-15,6-dichloro-N-(2,2-dimethoxyethyl)pyridin-3-amine
2933 39 99 1072-98-65-chloropyridin-2-amine
2933 39 99 298692-34-96-(chloroacetyl)pyridine-2-carboxylic acid
2933 39 99 550349-58-17-chloro-3-(6-methoxypyridin-3-yl)-N,N,5-trimethyl-4-oxo-4,5-dihydro-3H-pyridazino[4,5-b]indole-1-carboxamide
2933 39 99 414909-98-1benzyl 2-(4-fluoro-2-methylphenyl)-4-oxo-3,4-dihydropyridine-1(2H)-carboxylate
2933 39 99 56880-11-6ethyl [(3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl)acetate
2933 39 99 548797-97-3N-(2-{[(2S)-3-{[1-(4-chlorobenzyl)piperidin-4-yl]amino}-2-hydroxy-2-methylpropyl]oxy}-4-hydroxyphenyl)acetamide
2933 39 99 0-00-0N-[(S)-1-azabicyclo[2.2.2]oct-2-yl(phenyl)methyl]-2,6-dichloro-3-(trifluoromethyl)benzamide hydrochloride
2933 39 99 329003-65-8sodium hydrogen [1-hydroxy-1-phosphono-2-(pyridin-3-yl)ethyl]phosphonate hemipentahydrate
2933 49 10 417716-92-84-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide methanesulfonate
2933 49 90 503291-53-02-ethylbutyl (3S,4aS,6S,8aR)-6-[3-chloro-2-(1H-tetrazol-5-yl)phenoxy]decahydro-3-isoquinolinecarboxylate 4-methylbenzenesulfonate
2933 49 90 103733-32-0benzyl (3S)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-3-carboxylate hydrochloride
2933 49 90 503293-98-9(3S,4aS,6S,8aR)-6-hydroxy-2-(methoxycarbonyl)decahydroisoquinoline-3-carboxylic acid
2933 49 90 503290-66-2(3S,4aS,6S,8aR)-6-[3-chloro-2-(2H-tetrazol-5-yl)phenoxy]decahydro-3-isoquinolinecarboxylic acid hydrochloride
2933 49 90 134388-95-7(3S,4aS,8aR)-2-(methoxycarbonyl)-6-oxodecahydroisoquinoline-3-carboxylic acid – (1R)-1-phenylethanamine (1:1)
2933 49 90 868210-14-44-(4-{[(2S,4R)-4-[acetyl(4-chlorophenyl)amino]-2-methyl-3,4-dihydroquinolin-1(2H)-yl]carbonyl}phenoxy)-2,2-dimethylbutanoic acid
2933 49 90 00-00-0methyl 2-[(3R)-3-{3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl}-3-({[1-(hydroxymethyl)cyclopropyl]methyl}sulfanyl)propyl]benzoate hydrochloride
2933 49 90 848133-76-6N-(4-chloro-3-cyano-7-ethoxyquinolin-6-yl)acetamide
2933 59 95 869490-23-3(3,3-difluoropyrrolidin-1-yl){(2S,4S)-4-[4-(pyrimidin-2-yl)piperazin-1-yl]pyrrolidin-2-yl}methanone
2933 59 95 941685-40-1(3R)-3-cyclopentyl-3-[4-(7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile
2933 59 95 941678-49-5(3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile
2933 59 95 941685-41-2(3S)-3-cyclopentyl-3-[4-(7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile
2933 59 95 957187-34-7[(8R)-8-(3,5-difluorophenyl)-10-oxo-6,9-diazaspiro[4.5]dec-9-yl]acetic acid
2933 59 95 356058-42-9{2-[(4-fluorobenzyl)sulfanyl]-4-oxo-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidin-1-yl}acetic acid
2933 59 95 0-00-02,3-dihydroxy-2,3-bis(phenylcarbonyl)butanedioic acid – ethyl [(8R)-8-(3,5-difluorophenyl)-10-oxo-6,9-diazaspiro[4.5]dec-9-yl]acetate (1:1)
2933 59 95 90213-66-42,4-dichloro-7H-pyrrolo[2,3-d]pyrimidine
2933 59 95 3934-20-12,4-dichloropyrimidine
2933 59 95 451487-18-62-[(4-fluorobenzyl)sulfanyl]-1,5,6,7-tetrahydro-4H-cyclopenta[d]pyrimidin-4-one
2933 59 95 865758-96-92-[(6-chloro-3-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methyl]benzonitrile
2933 59 95 934815-71-12-[3-(6-{[2-(2,4-dichlorophenyl)ethyl]amino}-2-methoxypyrimidin-4-yl)phenyl]-2-methylpropanoic acid phosphate
2933 59 95 722543-31-92-{ethyl[3-({4-[(5-{2-[(3-fluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl)amino]quinazolin-7-yl}oxy)propyl]amino}ethyl dihydrogen phosphate
2933 59 95 1032066-96-82-amino-9-{(1S,3R,4S)-3-[(benzyloxy)methyl]-4-[dimethyl(phenyl)silyl]-2-methylidenecyclopentyl}-1,9-dihydro-6H-purin-6-one – methanesulfonate (2:1)
2933 59 95 540737-29-93-{(3R,4R)-4-methyl-3-[methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile 2-hydroxypropane-1,2,3-tricarboxylate
2933 59 95 1137917-12-43-{[6-(ethylsulfonyl)pyridin-3-yl]oxy}-5-{[(2S)-1-hydroxypropan-2-yl]oxy}benzoic acid – 1,4-diazabicyclo[2.2.2]octane (2:1)
2933 59 95 941685-39-83-cyclopentyl-3-[4-(7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile
2933 59 95 941685-27-44-(1H-pyrazol-4-yl)-7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidine
2933 59 95 1780-26-34,6-dichloro-2-methylpyrimidine
2933 59 95 145783-14-84,6-dichloro-5-nitro-2-(propylsulfanyl)pyrimidine
2933 59 95 3680-69-14-chloro-7H-pyrrolo[2,3-d]pyrimidine
2933 59 95 61379-64-44-cyclopentylpiperazin-1-amine
2933 59 95 55112-42-04-methylpiperazine-1-carbonyl chloride hydrochloride
2933 59 95 0-00-05-(benzylamino)-2-(3-methoxyphenyl)-7-(4-methylpiperazin-1-yl)[1,2,4]triazolo[1,5-a]quinoline-4-carbonitrile – (2E)-but-2-enedioate (2:1) hydrate
2933 59 95 55293-96-45,7-dimethyl[1,2,4]triazolo[1,5-a]pyrimidine-2-carbaldehyde
2933 59 95 179688-01-87-(benzyloxy)-6-methoxyquinazolin-4(3H)-one
2933 59 95 444731-74-2N-(2-chloropyrimidin-4-yl)-2,3-dimethyl-2H-indazol-6-amine
2933 59 95 0-00-0N-(5-fluoro-3-methyl-1H-indol-1-yl)-4-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2933 79 00 586414-48-4(-)-3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2H)-yl}-N,4-dimethylbenzamide
2933 79 00 425663-71-4(1S)-1-amino-3-methyl-1,3,4,5-tetrahydro-2H-3-benzazepin-2-one hydrochloride
2933 79 00 813452-14-1(4S)-1-[(2S,3S,11bS)-2-amino-9,10-dimethoxy-1,3,4,6,7,11b-hexahydro-2H-pyrido[2,1-a]isoquinolin-3-yl]-4-(fluoromethyl)pyrrolidin-2-one dihydrochloride
2933 79 00 5162-90-33-(2-oxo-1,2-dihydroquinolin-4-yl)alanine
2933 79 00 536760-29-93-chloro-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one
2933 79 00 4876-10-24-(bromomethyl)quinolin-2(1H)-one
2933 79 00 5057-12-54,6,7,8-tetrahydroquinoline-2,5(1H,3H)-dione
2933 79 00 54197-66-96-hydroxy-3,4-dihydroquinolin-2(1H)-one
2933 79 00 22246-18-07-hydroxy-3,4-dihydroquinolin-2(1H)-one
2933 79 00 536759-91-8ethyl 1-(4-methoxyphenyl)-6-(4-nitrophenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate
2933 79 00 503614-91-3ethyl 1-(4-methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate
2933 79 00 586379-61-5methyl 3-(4-hydroxy-6-methyl-2-oxopyridin-1(2H)-yl)-4-methylbenzoate
2933 99 80 709031-45-8(1S,3S,5S)-2-azabicyclo[3.1.0]hexane-3-carboxamide methanesulfonate
2933 99 80 649735-46-6(2R)-1-({4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl}oxy)propan-2-ol
2933 99 80 51077-14-6(2S)-1-(tert-butoxycarbonyl)azetidine-2-carboxylic acid
2933 99 80 631916-97-7(2S)-N-{4-[(Z)-amino(methoxyimino)methyl]benzyl}-1-{(2R)-2-[3-chloro-5-(difluoromethoxy)phenyl]-2-hydroxyethanoyl}azetidine-2-carboxamide – benzenesulphonic acid (1:1)
2933 99 80 80875-98-5(2S,3aS,7aS)-octahydro-1H-indole-2-carboxylic acid
2933 99 80 948846-40-0(2S,3S)-2,3-bis[(phenylcarbonyl)oxy]butanedioic acid – ethyl (3aR,6aR)-hexahydropyrrolo[3,4-b]pyrrole-5(1H)-carboxylate (1:1)
2933 99 80 1000164-36-2(5S,8S,11S,14S,17S,20S,23S,26S,29S,32S,35S,38S)-5-(3-amino-3-oxopropyl)-20-benzyl-23-[(2S)-butan-2-yl]-14,38-bis{4-[(tert-butoxycarbonyl)amino]butyl}-29-{[1-(tert-butoxycarbonyl)-1H-indol-3-yl]methyl}-17-(3-tert-butoxy-3-oxopropyl)-1-(1H-fluoren-9-yl)-8,11,26,41,41-pentamethyl-32-(2-methylpropyl)-3,6,9,12,15,18,21,24,27,30,33,36,39-tridecaoxo-35-(propan-2-yl)-2-oxa-4,7,10,13,16,19,22,25,28,31,34,37,40-tridecaazadotetracontan-42-oic acid
2933 99 80 22162-51-21-(2-nitrobenzyl)-1H-pyrrole-2-carbaldehyde
2933 99 80 35681-40-41-(propan-2-yl)-1,3-dihydro-2H-benzimidazol-2-one
2933 99 80 166170-15-61-(tert-butoxycarbonyl)-2-methyl-D-proline
2933 99 80 796967-16-31-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-5-methylphenyl)urea
2933 99 80 0-00-01-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-5-methylphenyl)urea hydrochloride
2933 99 80 444731-72-02,3-dimethyl-2H-indazol-6-amine
2933 99 80 19686-05-62,8-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
2933 99 80 912444-00-92-[(2R)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-4-carboxamide
2933 99 80 912445-36-42-[(2S)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-4-carboxamide dihydrochloride
2933 99 80 163457-23-63,3-difluoropyrrolidine hydrochloride
2933 99 80 239463-85-53-{5-[(2R)-2-aminopropyl]-7-cyano-2,3-dihydro-1H-indol-1-yl}propyl benzoate (2R,3R)-2,3-dihydroxybutanedioate
2933 99 80 55321-99-83-oxo-3,4-dihydropyrazine-2-carboxamide
2933 99 80 952490-01-64-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl 2,2-dimethylpropanoate
2933 99 80 942436-93-34-amino-8-(2,5-dimethoxyphenyl)-N-propylcinnoline-3-carboxamide
2933 99 80 942437-37-84-amino-8-(2-fluoro-6-methoxyphenyl)-N-propylcinnoline-3-carboxamide
2933 99 80 288385-88-64-fluoro-2-methyl-1H-indol-5-ol
2933 99 80 503293-47-85-(2-chloro-6-fluorophenyl)-2H-tetrazole
2933 99 80 73963-42-55-(4-chlorobutyl)-1-cyclohexyl-1H-tetrazole
2933 99 80 606143-52-65-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-N-(2-hydroxyethoxy)-1-methyl-1H-benzimidazole-6-carboxamide
2933 99 80 0-00-05-fluoro-1-(3-fluorobenzyl)-N-(1H-indol-5-yl)-1H-indole-2-carboxamide
2933 99 80 872206-47-85-methyl-4-oxo-1,4-dihydropyrrolo[2,1-f][1,2,4]triazin-6-yl 2,2-dimethylpropanoate
2933 99 80 259793-88-96-bromo-3-oxo-3,4-dihydropyrazine-2-carboxamide
2933 99 80 1137606-74-66-fluoro-3-oxo-3,4-dihydropyrazine-2-carbonitrile – N-cyclohexylcyclohexanamine (1:1)
2933 99 80 261953-36-06-iodo-1H-indazole
2933 99 80 80076-47-78,9-difluoro-5-methyl-1-oxo-6,7-dihydro-1H,5H-pyrido[3,2,1-ij]quinoline-2-carboxylic acid
2933 99 80 52602-39-89H-carbazol-4-ol
2933 99 80 145641-35-6benzyl (2S,3aR,7aS)-octahydro-1H-indole-2-carboxylate hydrochloride
2933 99 80 87269-87-2benzyl (2S,3aS,6aS)-octahydrocyclopenta[b]pyrrole-2-carboxylate hydrochloride
2933 99 80 1012065-72-3ethyl 2-amino-9,10-dimethoxy-1,6,7,11b-tetrahydro-4H-pyrido[2,1-a]isoquinoline-3-carboxylate
2933 99 80 131707-24-9ethyl 6-bromo-5-hydroxy-1-methyl-2-[(phenylsulfanyl)methyl]-1H-indole-3-carboxylate
2933 99 80 105152-95-2ethyl 7-(3-aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylate
2933 99 80 139481-44-0methyl 1-[(2′-cyanobiphenyl-4-yl)methyl]-2-ethoxy-1H-benzimidazole-7-carboxylate
2933 99 80 0-00-0methyl 1-tert-butyl-2-hydroxy-1H-pyrrolo[2,3-b]pyridine-3-carboxylate
2933 99 80 21688-11-9N2-[(benzyloxy)carbonyl]-L-glutaminyl-L-asparaginyl-S-benzyl-L-cysteinyl-L-prolyl-L-leucylglycinamide
2933 99 80 361440-67-7tert-butyl (1S,3S,5S)-3-carbamoyl-2-azabicyclo[3.1.0]hexane-2-carboxylate
2933 99 80 709031-38-9tert-butyl (2S)-2-carbamoyl-2,3-dihydro-1H-pyrrole-1-carboxylate
2933 99 80 709031-43-6tert-butyl [(1S)-2-[(1S,3S,5S)-3-cyano-2-azabicyclo[3.1.0]hex-2-yl]-1-(3-hydroxytricyclo[3.3.1.1(3,7)]dec-1-yl)-2-oxoethyl]carbamate
2933 49 90 936359-25-0methyl 2-((R)-3-(3-((E)-2-(7-chloroquinolin-2-yl)vinyl)phenyl)-3-(((1-(hydroxymethyl)cyclopropyl)methyl)sulfanyl)propyl)benzoate
2934 10 00 110130-88-6(2Z)-[(acetyloxy)imino](2-amino-1,3-thiazol-4-yl)ethanoic acid
2934 10 00 68672-66-2(2Z)-{[(1-tert-butoxy-2-methyl-1-oxopropan-2-yl)oxy]imino}[2-(tritylamino)-1,3-thiazol-4-yl]ethanoic acid
2934 10 00 291536-35-1(5Z)-5-(4-fluorobenzylidene)-1,3-thiazolidine-2,4-dione
2934 10 00 302964-24-52-amino-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide
2934 10 00 866920-24-33-[2-chloro-4-({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methoxy)phenyl]-1,2,4-oxadiazol-5(4H)-one
2934 10 00 752253-39-74-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(prop-2-yn-1-yl)-1,3-thiazol-2-amine
2934 10 00 914361-45-8L-lysine – {[(2R,3R)-3-[4-(4-cyanophenyl)-1,3-thiazol-2-yl]-2-(2,4-difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)butan-2-yl]oxy}methyl dihydrogen phosphate – ethanol (1:1:1)
2934 10 00 302964-08-5N-(2-chloro-6-methylphenyl)-2-[(6-chloro-2-methylpyrimidin-4-yl)amino]-1,3-thiazole-5-carboxamide
2934 10 00 127660-04-2sodium (2Z)-(2-amino-1,3-thiazol-4-yl)(hydroxyimino)ethanoate
2934 99 90 17381-54-3(1-benzothiophen-5-yl)acetic acid
2934 99 90 630100-90-2(1R)-1,2-anhydro-4-C-{(1E,3E)-4-[(1S,2S,3E,5R,6R,9R)-5-(1-carboxylato-4-cycloheptylpiperazin-2-yl)-6,9-dihydroxy-2,6-dimethyl-11-oxooxacyclododec-3-en-1-yl]penta-1,3-dien-1-yl}-3,5-dideoxy-1-[(2R,3S)-3-hydroxypentan-2-yl]-D-erythropentitol
2934 99 90 220099-91-2(2R)-3′H-spiro[4-azabicyclo[2.2.2]octane-2,2′-furo[2,3-b]pyridine]
2934 99 90 220100-81-2(2R)-3′H-spiro[4-azabicyclo[2.2.2]octane-2,2′-furo[2,3-b]pyridine] (S,S)-2,3-dihydroxybutanedioate
2934 99 90 161599-46-8(2R,3R,4R,5R)-2-(4-amino-5-fluoro-2-oxopyrimidin-1(2H)-yl)-2-fluoro-5-methyltetrahydrofuran-3,4-diyl diacetate
2934 99 90 690270-65-6(2R,3S,4R)-5-(4-amino-2-oxopyrimidin-1(2H)-yl)-2-azido-2-{[(2-methylpropanoyl)oxy]methyl}tetrahydrofuran-3,4-diyl bis(2-methylpropanoate) hydrochloride
2934 99 90 265121-04-8(3-{[(2R,3S)-2-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy}-3-(2-fluorophenyl)morpholin-4-yl]methyl}-5-oxo-2,5-dihydro-1H-1,2,4-triazol-1-yl)phosphonic acid – 1-deoxy-1-(methylamino)-D-glucitol (1:2)
2934 99 90 163680-80-6(3S)-10-[1-(acetylamino)cyclopropyl]-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7H-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxylic acid
2934 99 90 132335-46-7(3S)-N,N-dimethyl-3-(naphthalen-1-yloxy)-3-(thiophen-2-yl)propan-1-amine
2934 99 90 133413-70-4(3S,6R,9S,12R,15S,18R,21S,24R)-6,18-dibenzyl-4,10,12,16,22,24-hexamethyl-3,9,15,21-tetrakis(2-methylpropyl)-1,7,13,19-tetraoxa-4,10,16,22-tetraazacyclotetracosane-2,5,8,11,14,17,20,23-octone
2934 99 90 503068-36-8(5R)-3-(6-{2-[(2,6-dichlorobenzyl)oxy]ethoxy}hexyl)-5-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-1,3-oxazolidin-2-one
2934 99 90 452339-73-0(5R)-5-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-1,3-oxazolidin-2-one
2934 99 90 877130-28-4(6R)-6-cyclopentyl-6-[2-(2,6-diethylpyridin-4-yl)ethyl]-3-[(5,7-dimethyl[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methyl]-4-hydroxy-5,6-dihydro-2H-pyran-2-one
2934 99 90 132335-44-5(S)-3-(dimethylamino)-1-(thiophen-2-yl)propan-1-ol
2934 99 90 812647-80-6{(2R,3S,4R,5R)-2-azido-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-bis[(phenylcarbonyl)oxy]tetrahydrofuran-2-yl}methyl 3-chlorobenzoate
2934 99 90 00-00-01-(1-{4-[2-(4-fluorophenyl)-1,3-dioxolan-2-yl]butyl}-1,2,3,6-tetrahydropyridin-4-yl)-1,3-dihydro-2H-benzimidazol-2-one
2934 99 90 1029716-44-61-(1-ethoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole
2934 99 90 165172-60-11-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]-5-methylpyrimidine-2,4(1H,3H)-dione – 1-methylpyrrolidin-2-one (1:1)
2934 99 90 519187-97-41-[3-(2-benzo[b]thien-5-ylethoxy)propyl]-3-azetidinol – (2Z)-2-butenedioate (1:1)
2934 99 90 127000-90-21-{[(2R,3S)-2-(2,4-difluorophenyl)-3-methyloxiran-2-yl]methyl}-1H-1,2,4-triazole
2934 99 90 710281-33-72-({[(1R,3S)-3-{[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}cyclohexyl]oxy}methyl)-6-methylbenzoic acid
2934 99 90 96803-30-42-(1-benzothiophen-5-yl)ethanol
2934 99 90 913695-00-82-[({4-[(2,2-dimethyl-1,3-dioxan-5-yl)methoxy]-3,5-dimethylpyridin-2-yl}methyl)sulfinyl]-1Hbenzimidazole, sodium salt (1:1)
2934 99 90 376608-74-12-{[(3aR,4S,6R,6aS)-6-{[5-amino-6-chloro-2-(propylsulfanyl)pyrimidin-4-yl]amino}-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl]oxy}ethanol
2934 99 90 474554-48-82-bromo-1-[3-tert-butyl-4-methoxy-5-(morpholin-4-yl)phenyl]ethanone
2934 99 90 530141-72-13-(5-{[4-(cyclopentyloxy)-2-hydroxyphenyl]carbonyl}-2-[(3-hydroxy-1,2-benzoxazol-6-yl)methoxy]phenyl)propanoic acid
2934 99 90 519188-55-73-[2-(1-benzothiophen-5-yl)ethoxy]-1-(3-hydroxyazetidin-1-yl)propan-1-one
2934 99 90 519188-42-23-[2-(1-benzothiophen-5-yl)ethoxy]propionic acid
2934 99 90 753015-42-83-{(E)-2-[(3R)-pyrrolidin-3-yl]ethenyl}-5-(tetrahydro-2H-pyran-4-yloxy)pyridine
2934 99 90 26638-53-93-chloro-6-methyldibenzo[c,f][1,2]thiazepin-11(6H)-one 5,5-dioxide
2934 99 90 499785-81-83-oxo-4-(2,3,5-tri-O-acetyl-β-D-ribofuranosyl)-3,4-dihydropyrazine-2-carboxamide
2934 99 90 356782-84-83-oxo-4-(β-D-ribofuranosyl)-3,4-dihydropyrazine-2-carboxamide
2934 99 90 6504-57-04-[3-hydroxy-3-phenyl-3-(thiophen-2-yl)propyl]-4-methylmorpholin-4-ium methyl sulfate
2934 99 90 871484-32-14-[4-({3-[(4-deoxy-4-fluoro-b-D-glucopyranosyl)oxy]-5-(propan-2-yl)-1H-pyrazol-4-yl}methyl)phenyl]-N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]butanamide
2934 99 90 166964-09-64-chloro-3-methyl-1,2-oxazol-5-amine
2934 99 90 655233-39-34-nitrobenzyl(6R,7R)-7-amino-8-oxo-3-[(2S)-tetrahydrofuran-2-yl]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate hydrochloride
2920 90 85 89729-09-95,7-dioxa-6-thiaspiro[2.5]octane-6-oxide
2934 99 90 388082-75-55-[4-[[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]amino]-6-quinazolinyl]-2-furancarboxaldehyde – 4-methylbenzenesulfonate (1:1)
2934 99 90 4923-87-95-bromo-1-benzothiophene
2934 99 90 947408-95-96-(bromomethyl)-2-triphenylmethyl-1,2-benzisoxazol-3(2H)-one
2934 99 90 947408-94-86-methyl-2-trityl-1,2-benzoxazol-3(2H)-one
2934 99 90 67978-05-6diphenylmethyl(2R)-3-methyl-2-[(1R,5S)-3-(4-methylphenyl)-7-oxo-4-oxa-2,6-diazabicyclo[3.2.0]hept-2-en-6-yl]but-3-enoate
2934 99 90 1001859-46-6DNA (synthetic plasmid vector pCOR human interferon beta signal peptide fusion protein with 21-154-human acidic fibroblast growth factor-specifying)
2934 99 90 665058-78-6DNA, d(T-sp-C-G-sp-T-sp-C-G-sp-T-sp-T-sp-T-sp-T-sp-G-sp-A-sp-C-G-sp-T-sp-T-sp-T-sp-T-sp-Gsp-T-sp-C-G-sp-T-sp-T)
2934 99 90 923591-06-4methyl (5R,7S,10S)-10-tert-butyl-15,15-dimethyl-3,9,12-trioxo-6,7,9,10,11,12,14,15,16,17,18,19-dodecahydro-1H,5H-2,23:5,8-dimethano-4,13,2,8,11-benzodioxatriazacyclohenicosine-7(3H)-carboxylate
2934 99 90 59337-92-7methyl 3-(chlorosulfonyl)thiophene-2-carboxylate
2934 99 90 947409-01-0methyl 3-[5-[4-(cyclopentyloxy)-2-hydroxybenzoyl]-2-[(2-triphenylmethyl-1,2-benzisoxazol-3(2H)-on-6-yl)methoxy]phenyl]propionate
2934 99 90 85006-31-1methyl 3-amino-4-methylthiophene-2-carboxylate
2934 99 90 893428-72-3N-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methyl-1-piperazinyl)ethoxy]-5-[(tetrahydro-2H-pyran-4-yl)oxy]-4-quinazolinamine – (2E)-2-butenedioate (1:2)
2934 99 90 390800-88-1N,N′,N′′-(boroxin-2,4,6-triyltris{[(1S)-3-methylbutane-1,1-diyl]imino[(2S)-1-oxo-3-phenylpropane-1,2-diyl]})tripyrazine-2-carboxamide
2934 99 90 112913-94-7N-{[4-(4-fluorobenzyl)morpholin-2-yl]methyl}acetamide
2934 99 90 120788-03-6S-[(1R,3S)-1-oxidotetrahydrothiophen-3-yl] ethanethioate
2935 00 90 1198178-65-2(1R,2R)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethylcyclopropanaminium 4-methylbenzenesulfonate
2935 00 90 39570-96-2(2R)-3-(benzylsulfanyl)-N-[(2S)-1-{[(2S,3S)-1-hydrazinyl-3-methyl-1-oxopentan-2-yl]amino}-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-2-{[(4-methylphenyl)sulfonyl]amino}propanamide
2935 00 90 24310-36-91-[(4-methylphenyl)sulfonyl]-1,2,3,4-tetrahydro-5H-1-benzazepin-5-one
2935 00 90 0-00-02-(cyclohexylmethyl)-N-{2-[(2S)-1-methylpyrrolidin-2-yl]ethyl}-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide di[(2E)-but-2-enedioate] hydrate
2935 00 90 941690-55-73-[(methylsulfonyl)amino]-2-phenyl-N-[(1S)-1-phenylpropyl]quinoline-4-carboxamide
2935 00 90 6973-09-75-amino-2-methylbenzenesulfonamide
2935 00 90 193686-76-97-chloro-1-[(4-methylphenyl)sulfonyl]-1,2,3,4-tetrahydro-5H-1-benzazepin-5-one
2935 00 90 123664-84-6N-(5-methoxy-2-phenoxyphenyl)methanesulfonamide
2935 00 90 149457-03-4N-[4-(N-formylglycyl)-5-hydroxy-2-phenoxyphenyl]methanesulfonamide
2935 00 90 149456-98-4N-[4-(N-formylglycyl)-5-methoxy-2-phenoxyphenyl]methanesulfonamide
2935 00 90 141450-48-8N-{2-[(4-hydroxyphenyl)amino]pyridin-3-yl}-4-methoxybenzenesulfonamide hydrochloride
2935 00 90 289042-10-0N-{5-[(diphenylphosphoryl)methyl]-4-(4-fluorophenyl)-6-(propan-2-yl)pyrimidin-2-yl}-N-methylmethanesulfonamide
2939 99 00 7689-03-4(4S)-4-ethyl-4-hydroxy-1H-pyrano[3′,4′:6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione
2939 99 00 477-29-2colchicoside
2940 00 00 604-69-31,2,3,4,6-penta-O-acetyl-β-D-glucopyranose
2940 00 00 647834-15-92-(4-methoxybenzyl)thiophen-3-yl β-D-glucopyranoside
2941 90 00 76610-92-9(6R,7R)-7-({N-[(4-ethyl-2,3-dioxopiperazin-1-yl)carbonyl]-D-threonyl}amino)-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
3907 20 99 913976-27-9poly(oxy-1,2-ethanediyl), α-hydro-ω-methoxy, diester with 21N6, 21′N6-[[(N2, N6-dicarboxy-L-lysyl-β-alanyl)imino]bis(1-oxo-2, 1-ethanediyl)]bis[N-acetylglycyl-L-leucyl-L-tyrosyl-L-alanyl-L-cysteinyl-L-histidyl-L-methionylglycyl-L-prolyl-L-isoleucyl-L-threonyl-3-(1-naphthalenyl)-L-alanyl-L-valyl-L-cysteinyl-L-glutaminyl-L-prolyl-L-leucyl-L-arginyl-N-methylglycyl-L-lysinamide] cyclic (6→15), (6′→15′) bis(disulfide)

Annex IV

List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be withdrawn from the list of products receiving duty-free treatment included in Annex 6 to Annex I to Regulation (EEC) No 2658/87 due to their transfer to the list of products receiving duty-free treatment included in Annex 3 to Annex I to Regulation (EEC) No 2658/87

CN codeCAS RNName

2915 39 00

2937 29 00

7753-60-8

17-alpha-hydroxy-3,20-dioxopregna-4,9(11)-diene-21-yl acetate

see anecortave (INN)

2920 90 85 163133-43-5

4-(nitrooxy)butyl (2S)-2-(6-methoxy-2-naphthyl) propanoate

see naproxcinod (INN)

2924 29 98 194085-75-1

2-(2-chlorophenyl)-2-hydroxyethyl carbamate

see carisbamate (INN)

2933 39 99 103129-82-4

3-ethyl 5-methyl 2-[(2-aminoethoxy)methyl]-4-(2-chlorophenyl)-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate

see levamlodipine (INN)

2933 39 99 319460-85-0

N-methyl-2-{[3-((E)-2-pyridin-2-ylvinyl)-1H-indazol-6-yl]sulfanyl}benzamide

see axitinib (INN)

2934 10 00 302962-49-8

N-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)thiazole-5-carboxamide

see dasatinib (INN)

2934 99 90 143491-57-0

(2R,5S)-4-amino-5-fluoro-1-[2-(hydroxymethyl)-1,3-oxathiolan-5-yl]pyrimidin-2(1H)-one

see emtricitabine(INN)

2934 99 90 98819-76-2

(2S)-2-[(S)-(2-ethoxyphenoxy)phenylmethyl]morpholine

see esreboxetine (INN)

2934 99 90 475479-34-6

(2S)-2-methoxy-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]-1-benzothiophen-7-yl}propanoic acid

see aleglitazar (INN)

2934 99 90 377727-87-2

2-(2-furyl)-7-(2-{4-[4-(2-methoxyethoxy)phenyl] piperazin-1-yl}ethyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[2,3-c]pyrimidin-5-amine

see preladenant (INN)

2934 99 90 189003-92-7

2-{7-fluoro-2-oxo-4-[2-(4-thieno[3,2-c]pyridin-4-ylpiperazin-1-yl)ethyl]quinolin-1(2H)-yl}acetamide

see trelanserin (INN)

2934 99 90 134379-77-4

4-amino-5-fluoro-1-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]pyrimidin-2(1H)-one

see dexelvucitabine (INN)

2934 99 90 518048-05-0

potassium 4-[N-(2-fluorobenzyl)carbamoyl]-1-methyl-2-[1-methyl-1-(5-methyl-1,3,4-oxadiazole-2-carboxamido)ethyl]-6-oxo-1,6-dihydropyrimidine-5-olate

see raltegravir (INN)

2935 00 90 170569-88-7

4-[5-(4-fluorophenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzene-1-sulfonamide

see mavacoxib (INN)

2935 00 90 186497-07-4

N-(3-methoxy-5-methylpyrazin-2-yl)-2-[4-(1,3,4-oxadiazol-2-yl)phenyl]pyridine-3-sulfonamide

see zibotentan (INN)